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authFullName_s : Étienne Billard

Discovery of New Allosteric Modulators of the Urotensinergic System through Substitution of the Urotensin II-Related Peptide (URP) Phenylalanine Residue

Étienne Billard , Terence Hébert , David Chatenet
Journal of Medicinal Chemistry, 2018, 61 (19), pp.8707-8716. ⟨10.1021/acs.jmedchem.8b00789⟩
Journal articles pasteur-02133248v1

Functional Selectivity Revealed by N-Methylation Scanning of Human Urotensin II and Related Peptides

Francesco Merlino , Étienne Billard , Ali M. Yousif , Salvatore Di Maro , Diego Brancaccio , et al.
Journal of Medicinal Chemistry, 2019, 62 (3), pp.1455-1467. ⟨10.1021/acs.jmedchem.8b01601⟩
Journal articles pasteur-02136107v1

Urotensin II((4-11)) Azasulfuryl Peptides: Synthesis and Biological Activity.

Francesco Merlino , Ali M Yousif , Étienne Billard , Julien Dufour-Gallant , Stéphane Turcotte , et al.
Journal of Medicinal Chemistry, 2016, 59 (10), pp.4740-52. ⟨10.1021/acs.jmedchem.6b00108⟩
Journal articles pasteur-01351481v1

Design, Synthesis, and Biological Assessment of Biased Allosteric Modulation of the Urotensin II Receptor Using Achiral 1,3,4-Benzotriazepin-2-one Turn Mimics

Antoine Douchez , Étienne Billard , Terence Hébert , David Chatenet , William Lubell
Journal of Medicinal Chemistry, 2017, 60 (23), pp.9838 - 9859. ⟨10.1021/acs.jmedchem.7b01525⟩
Journal articles pasteur-01688987v1
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Design of a peptidic inhibitor that targets the dimer interface of a prototypic galectin.

Maria Claudia Vladoiu , Marilyne Labrie , Myriam Létourneau , Philippe Egesborg , Donald Gagné , et al.
Oncotarget, 2015, 6 (38), pp.40970-80. ⟨10.18632/oncotarget.5403⟩
Journal articles pasteur-01352682v1

Urotensin core mimics that modulate the biological activity of urotensin-II related peptide but not urotensin-II.

Martin Strack , Étienne Billard , David Chatenet , William D Lubell
Bioorganic and Medicinal Chemistry Letters, 2017, 27 (15), pp.3412-3416. ⟨10.1016/j.bmcl.2017.05.088⟩
Journal articles pasteur-01574618v1

New directions for urotensin II receptor ligands

Etienne Billard , Étienne Billard , Mustapha Iddir , Hassan Nassour , Laura Lee-Gosselin , et al.
Peptide Science, 2018, 111 (1), pp.e24056. ⟨10.1002/pep2.24056⟩
Journal articles pasteur-02133250v1