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Identification of a novel quinoline-based DNA demethylating compound highly potent in cancer cells
Clemens Zwergel
,
Michael Schnekenburger
,
Federica Sarno
,
Cecilia Battistelli
,
Maria Cristina Manara
,
et al.
Journal articles
hal-02383678v1
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Novel benzofuran-chromone and -coumarin derivatives: synthesis and biological activity in K562 human leukemia cells
Clemens Zwergel
,
Sergio Valente
,
Angela Salvato
,
Zhanjie Xu
,
Oualid Talhi
,
et al.
Journal articles
hal-01494094v1
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Novel Quinoline Compounds Active in Cancer Cells through Coupled DNA Methyltransferase Inhibition and Degradation
Clemens Zwergel
,
Rossella Fioravanti
,
Giulia Stazi
,
Federica Sarno
,
Cecilia Battistelli
,
et al.
Journal articles
pasteur-03026533v1
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A Quinoline-Based DNA Methyltransferase Inhibitor as a Possible Adjuvant in Osteosarcoma Therapy
Maria Cristina Manara
,
Sergio Valente
,
Camilla Cristalli
,
Giordano Nicoletti
,
Lorena Landuzzi
,
et al.
Journal articles
hal-02383680v1
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Novel reversible monoamine oxidase A inhibitors: highly potent and selective 3-(1H-pyrrol-3-yl)-2-oxazolidinones.
Sergio Valente
,
Stefano Tomassi
,
Giampiero Tempera
,
Stefania Saccoccio
,
Enzo Agostinelli
,
et al.
Journal articles
pasteur-00980200v1
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Interplay among nucleosomal DNA, histone tails, and corepressor CoREST underlies LSD1-mediated H3 demethylation.
Simona Pilotto
,
Valentina Speranzini
,
Marcello Tortorici
,
Dominique Durand
,
Alexander Fish
,
et al.
Proceedings of the National Academy of Sciences of the United States of America, 2015, 112 (9), pp.2752-7. ⟨10.1073/pnas.1419468112⟩
Journal articles
hal-01448118v1
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Identification of novel quinazoline derivatives as potent antiplasmodial agents
Anne Bouchut
,
Dante Rotili
,
Christine Pierrot
,
Sergio Valente
,
Sophia Lafitte
,
et al.
Journal articles
pasteur-03036828v1
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Novel 3,5-bis(bromohydroxybenzylidene)piperidin-4-ones as coactivator-associated arginine methyltransferase 1 inhibitors: enzyme selectivity and cellular activity.
Donghang Cheng
,
Sergio Valente
,
Sabrina Castellano
,
Gianluca Sbardella
,
Roberto Di Santo
,
et al.
Journal articles
pasteur-00968654v1
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Reactivity of 4-Vinyl-2H-1-benzopyran-2-ones in Diels-Alder Cycloaddition Reactions: Access to Coumarin-Based Polycycles with Cdc25 Phosphatase-Inhibiting Activity
Sergio Valente
,
Zhanjie Xu
,
Emilie Bana
,
Clemens Zwergel
,
Antonello Mai
,
et al.
Journal articles
istex
hal-01494085v1
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Combined HAT/EZH2 modulation leads to cancer-selective cell death
Francesca Petraglia
,
Abhishek Singh
,
Vincenzo Carafa
,
Angela Nebbioso
,
Mariarosaria Conte
,
et al.
Journal articles
hal-01873834v1
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Specific activity of class II histone deacetylases in human breast cancer cells.
Vanessa Duong
,
Caroline Bret
,
Lucia Altucci
,
Antonello Mai
,
Céline Duraffourd
,
et al.
Journal articles
inserm-00351047v1
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Novel inhibitors of human histone deacetylases: Design, synthesis and bioactivity of 3-alkenoylcoumarines
Carole Seidel
,
Michael Schnekenburger
,
Clemens Zwergel
,
François Gaascht
,
Antonello Mai
,
et al.
Journal articles
hal-01494600v1
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Targeting RAGE prevents muscle wasting and prolongs survival in cancer cachexia
Alessandra Renzini
,
Nicoletta Marroncelli
,
Giorgia Cavioli
,
Silvia Di Francescantonio
,
Laura Forcina
,
et al.
Journal articles
hal-03714907v1
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Selective class II HDAC inhibitors impair myogenesis by modulating the stability and activity of HDAC-MEF2 complexes.
Angela Nebbioso
,
Fabio Manzo
,
Marco Miceli
,
Mariarosaria Conte
,
Lucrezia Manente
,
et al.
Journal articles
inserm-00420167v1
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Selective Non-nucleoside Inhibitors of Human DNA Methyltransferases Active in Cancer Including in Cancer Stem Cells
Sergio Valente
,
Yiwei Liu
,
Michael Schnekenburger
,
Clemens Zwergel
,
Sandro Cosconati
,
et al.
Journal articles
hal-01494552v1
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Identification of PR-SET7 and EZH2 selective inhibitors inducing cell death in human leukemia U937 cells.
Sergio Valente
,
Ilaria Lepore
,
Carmela Dell'Aversana
,
Maria Tardugno
,
Sabrina Castellano
,
et al.
Journal articles
pasteur-00968696v1
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New Insights on the Mechanism of Quinoline-based DNA Methyltransferase Inhibitors
Christina Gros
,
Laurence Fleury
,
Virginie Nahoum
,
Céline Faux
,
Sergio Valente
,
et al.
Journal articles
hal-03002969v1
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