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Phenylpyrazolo[1,5-a]quinazolin-5(4H)-one: a suitable scaffold for the development of noncamptothecin topoisomerase I (Top1) inhibitors.
Sabrina Taliani
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Isabella Pugliesi
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Elisabetta Barresi
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Silvia Salerno
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Christophe Marchand
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et al.
Journal articles
pasteur-00968854v1
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Quinolinonyl Non-Diketo Acid Derivatives as Inhibitors of HIV-1 Ribonuclease H and Polymerase Functions of Reverse Transcriptase
Antonella Messore
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Angela Corona
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Valentina Noemi Madia
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Francesco Saccoliti
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Valeria Tudino
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et al.
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hal-03831904v1
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New nitrogen containing substituents at the indole-2-carboxamide yield high potent and broad spectrum indolylarylsulfone HIV-1 non-nucleoside reverse transcriptase inhibitors.
Giuseppe La Regina
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Antonio Coluccia
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Andrea Brancale
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Francesco Piscitelli
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Valeria Famiglini
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et al.
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pasteur-00969585v1
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Selective Non-nucleoside Inhibitors of Human DNA Methyltransferases Active in Cancer Including in Cancer Stem Cells
Sergio Valente
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Yiwei Liu
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Michael Schnekenburger
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Clemens Zwergel
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Sandro Cosconati
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et al.
Journal articles
hal-01494552v1
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Properly Substituted Analogues of BIX-01294 Lose Inhibition of G9a Histone Methyltransferase and Gain Selective Anti-DNA Methyltransferase 3A Activity
Dante Rotili
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Domenico Tarantino
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Biagina Marrocco
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Christina Gros
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Véronique Masson
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et al.
Journal articles
pasteur-03182293v1
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