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New nucleotide-competitive non-nucleoside inhibitors of terminal deoxynucleotidyl transferase: discovery, characterization, and crystal structure in complex with the target.

Roberta Costi , Giuliana Cuzzucoli Crucitti , Luca Pescatori , Antonella Messore , Luigi Scipione , et al.
Journal of Medicinal Chemistry, 2013, 56 (18), pp.7431-41. ⟨10.1021/jm4010187⟩
Journal articles pasteur-00968827v1
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New nitrogen containing substituents at the indole-2-carboxamide yield high potent and broad spectrum indolylarylsulfone HIV-1 non-nucleoside reverse transcriptase inhibitors.

Giuseppe La Regina , Antonio Coluccia , Andrea Brancale , Francesco Piscitelli , Valeria Famiglini , et al.
Journal of Medicinal Chemistry, 2012, 55 (14), pp.6634-8. ⟨10.1021/jm300477h⟩
Journal articles pasteur-00969585v1
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Effects of polyphenol compounds on influenza A virus replication and definition of their mechanism of action.

Rossella Fioravanti , Ignacio Celestino , Roberta Costi , Giuliana Cuzzucoli Crucitti , Luca Pescatori , et al.
Bioorganic and Medicinal Chemistry, 2012, 20 (16), pp.5046-52. ⟨10.1016/j.bmc.2012.05.062⟩
Journal articles pasteur-00968715v1
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6-(1-Benzyl-1H-pyrrol-2-yl)-2,4-dioxo-5-hexenoic acids as dual inhibitors of recombinant HIV-1 integrase and ribonuclease H, synthesized by a parallel synthesis approach.

Roberta Costi , Mathieu Métifiot , Francesca Esposito , Giuliana Cuzzucoli Crucitti , Luca Pescatori , et al.
Journal of Medicinal Chemistry, 2013, 56 (21), pp.8588-98. ⟨10.1021/jm401040b⟩
Journal articles pasteur-00968870v1
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Phenylpyrazolo[1,5-a]quinazolin-5(4H)-one: a suitable scaffold for the development of noncamptothecin topoisomerase I (Top1) inhibitors.

Sabrina Taliani , Isabella Pugliesi , Elisabetta Barresi , Silvia Salerno , Christophe Marchand , et al.
Journal of Medicinal Chemistry, 2013, 56 (18), pp.7458-62. ⟨10.1021/jm400932c⟩
Journal articles pasteur-00968854v1

Quinolinonyl Non-Diketo Acid Derivatives as Inhibitors of HIV-1 Ribonuclease H and Polymerase Functions of Reverse Transcriptase

Antonella Messore , Angela Corona , Valentina Noemi Madia , Francesco Saccoliti , Valeria Tudino , et al.
Journal of Medicinal Chemistry, 2021, 64 (12), pp.8579-8598. ⟨10.1021/acs.jmedchem.1c00535⟩
Journal articles hal-03831904v1

Functional Selectivity Revealed by N-Methylation Scanning of Human Urotensin II and Related Peptides

Francesco Merlino , Étienne Billard , Ali M. Yousif , Salvatore Di Maro , Diego Brancaccio , et al.
Journal of Medicinal Chemistry, 2019, 62 (3), pp.1455-1467. ⟨10.1021/acs.jmedchem.8b01601⟩
Journal articles pasteur-02136107v1
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Combined HAT/EZH2 modulation leads to cancer-selective cell death

Francesca Petraglia , Abhishek Singh , Vincenzo Carafa , Angela Nebbioso , Mariarosaria Conte , et al.
Oncotarget, 2018, 9 (39), pp.25630-25646. ⟨10.18632/oncotarget.25428⟩
Journal articles hal-01873834v1

Selective Non-nucleoside Inhibitors of Human DNA Methyltransferases Active in Cancer Including in Cancer Stem Cells

Sergio Valente , Yiwei Liu , Michael Schnekenburger , Clemens Zwergel , Sandro Cosconati , et al.
Journal of Medicinal Chemistry, 2014, 57 (3), pp.701-713. ⟨10.1021/jm4012627⟩
Journal articles hal-01494552v1
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Properly Substituted Analogues of BIX-01294 Lose Inhibition of G9a Histone Methyltransferase and Gain Selective Anti-DNA Methyltransferase 3A Activity

Dante Rotili , Domenico Tarantino , Biagina Marrocco , Christina Gros , Véronique Masson , et al.
PLoS ONE, 2014, 9 (5), pp.e96941. ⟨10.1371/journal.pone.0096941⟩
Journal articles pasteur-03182293v1
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Identification of PR-SET7 and EZH2 selective inhibitors inducing cell death in human leukemia U937 cells.

Sergio Valente , Ilaria Lepore , Carmela Dell'Aversana , Maria Tardugno , Sabrina Castellano , et al.
Biochimie, 2012, 94 (11), pp.2308-13. ⟨10.1016/j.biochi.2012.06.003⟩
Journal articles pasteur-00968696v1
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The effect of d-amino acid substitution on the selectivity of temporin L towards target cells: identification of a potent anti-Candida peptide.

Paolo Grieco , Alfonso Carotenuto , Luigia Auriemma , Maria Rosaria Saviello , Pietro Campiglia , et al.
BBA - Biochimica et Biophysica Acta, 2013, 1828 (2), pp.652-60. ⟨10.1016/j.bbamem.2012.08.027⟩
Journal articles pasteur-00968523v1