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New nucleotide-competitive non-nucleoside inhibitors of terminal deoxynucleotidyl transferase: discovery, characterization, and crystal structure in complex with the target.
Roberta Costi
,
Giuliana Cuzzucoli Crucitti
,
Luca Pescatori
,
Antonella Messore
,
Luigi Scipione
,
et al.
Journal articles
pasteur-00968827v1
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New nitrogen containing substituents at the indole-2-carboxamide yield high potent and broad spectrum indolylarylsulfone HIV-1 non-nucleoside reverse transcriptase inhibitors.
Giuseppe La Regina
,
Antonio Coluccia
,
Andrea Brancale
,
Francesco Piscitelli
,
Valeria Famiglini
,
et al.
Journal articles
pasteur-00969585v1
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Effects of polyphenol compounds on influenza A virus replication and definition of their mechanism of action.
Rossella Fioravanti
,
Ignacio Celestino
,
Roberta Costi
,
Giuliana Cuzzucoli Crucitti
,
Luca Pescatori
,
et al.
Journal articles
pasteur-00968715v1
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6-(1-Benzyl-1H-pyrrol-2-yl)-2,4-dioxo-5-hexenoic acids as dual inhibitors of recombinant HIV-1 integrase and ribonuclease H, synthesized by a parallel synthesis approach.
Roberta Costi
,
Mathieu Métifiot
,
Francesca Esposito
,
Giuliana Cuzzucoli Crucitti
,
Luca Pescatori
,
et al.
Journal articles
pasteur-00968870v1
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Phenylpyrazolo[1,5-a]quinazolin-5(4H)-one: a suitable scaffold for the development of noncamptothecin topoisomerase I (Top1) inhibitors.
Sabrina Taliani
,
Isabella Pugliesi
,
Elisabetta Barresi
,
Silvia Salerno
,
Christophe Marchand
,
et al.
Journal articles
pasteur-00968854v1
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Quinolinonyl Non-Diketo Acid Derivatives as Inhibitors of HIV-1 Ribonuclease H and Polymerase Functions of Reverse Transcriptase
Antonella Messore
,
Angela Corona
,
Valentina Noemi Madia
,
Francesco Saccoliti
,
Valeria Tudino
,
et al.
Journal articles
hal-03831904v1
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Functional Selectivity Revealed by N-Methylation Scanning of Human Urotensin II and Related Peptides
Francesco Merlino
,
Étienne Billard
,
Ali M. Yousif
,
Salvatore Di Maro
,
Diego Brancaccio
,
et al.
Journal articles
pasteur-02136107v1
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Combined HAT/EZH2 modulation leads to cancer-selective cell death
Francesca Petraglia
,
Abhishek Singh
,
Vincenzo Carafa
,
Angela Nebbioso
,
Mariarosaria Conte
,
et al.
Journal articles
hal-01873834v1
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Selective Non-nucleoside Inhibitors of Human DNA Methyltransferases Active in Cancer Including in Cancer Stem Cells
Sergio Valente
,
Yiwei Liu
,
Michael Schnekenburger
,
Clemens Zwergel
,
Sandro Cosconati
,
et al.
Journal articles
hal-01494552v1
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Properly Substituted Analogues of BIX-01294 Lose Inhibition of G9a Histone Methyltransferase and Gain Selective Anti-DNA Methyltransferase 3A Activity
Dante Rotili
,
Domenico Tarantino
,
Biagina Marrocco
,
Christina Gros
,
Véronique Masson
,
et al.
Journal articles
pasteur-03182293v1
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Identification of PR-SET7 and EZH2 selective inhibitors inducing cell death in human leukemia U937 cells.
Sergio Valente
,
Ilaria Lepore
,
Carmela Dell'Aversana
,
Maria Tardugno
,
Sabrina Castellano
,
et al.
Journal articles
pasteur-00968696v1
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The effect of d-amino acid substitution on the selectivity of temporin L towards target cells: identification of a potent anti-Candida peptide.
Paolo Grieco
,
Alfonso Carotenuto
,
Luigia Auriemma
,
Maria Rosaria Saviello
,
Pietro Campiglia
,
et al.
Journal articles
pasteur-00968523v1
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