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Phenylpyrazolo[1,5-a]quinazolin-5(4H)-one: a suitable scaffold for the development of noncamptothecin topoisomerase I (Top1) inhibitors.

Sabrina Taliani , Isabella Pugliesi , Elisabetta Barresi , Silvia Salerno , Christophe Marchand , et al.
Journal of Medicinal Chemistry, 2013, 56 (18), pp.7458-62. ⟨10.1021/jm400932c⟩
Journal articles pasteur-00968854v1

Quinolinonyl Non-Diketo Acid Derivatives as Inhibitors of HIV-1 Ribonuclease H and Polymerase Functions of Reverse Transcriptase

Antonella Messore , Angela Corona , Valentina Noemi Madia , Francesco Saccoliti , Valeria Tudino , et al.
Journal of Medicinal Chemistry, 2021, 64 (12), pp.8579-8598. ⟨10.1021/acs.jmedchem.1c00535⟩
Journal articles hal-03831904v1
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New nucleotide-competitive non-nucleoside inhibitors of terminal deoxynucleotidyl transferase: discovery, characterization, and crystal structure in complex with the target.

Roberta Costi , Giuliana Cuzzucoli Crucitti , Luca Pescatori , Antonella Messore , Luigi Scipione , et al.
Journal of Medicinal Chemistry, 2013, 56 (18), pp.7431-41. ⟨10.1021/jm4010187⟩
Journal articles pasteur-00968827v1
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Effects of polyphenol compounds on influenza A virus replication and definition of their mechanism of action.

Rossella Fioravanti , Ignacio Celestino , Roberta Costi , Giuliana Cuzzucoli Crucitti , Luca Pescatori , et al.
Bioorganic and Medicinal Chemistry, 2012, 20 (16), pp.5046-52. ⟨10.1016/j.bmc.2012.05.062⟩
Journal articles pasteur-00968715v1
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6-(1-Benzyl-1H-pyrrol-2-yl)-2,4-dioxo-5-hexenoic acids as dual inhibitors of recombinant HIV-1 integrase and ribonuclease H, synthesized by a parallel synthesis approach.

Roberta Costi , Mathieu Métifiot , Francesca Esposito , Giuliana Cuzzucoli Crucitti , Luca Pescatori , et al.
Journal of Medicinal Chemistry, 2013, 56 (21), pp.8588-98. ⟨10.1021/jm401040b⟩
Journal articles pasteur-00968870v1
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Novel 3,5-bis(bromohydroxybenzylidene)piperidin-4-ones as coactivator-associated arginine methyltransferase 1 inhibitors: enzyme selectivity and cellular activity.

Donghang Cheng , Sergio Valente , Sabrina Castellano , Gianluca Sbardella , Roberto Di Santo , et al.
Journal of Medicinal Chemistry, 2011, 54 (13), pp.4928-32. ⟨10.1021/jm200453n⟩
Journal articles pasteur-00968654v1
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Pharmacophore assessment through 3-D QSAR: evaluation of the predictive ability on new derivatives by the application on a series of antitubercular agents.

Laura Friggeri , Flavio Ballante , Rino Ragno , Ira Musmuca , Daniela de Vita , et al.
Journal of Chemical Information and Modeling, 2013, 53 (6), pp.1463-74. ⟨10.1021/ci400132q⟩
Journal articles pasteur-00968810v1
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Synthesis and antifungal activity of a new series of 2-(1H-imidazol-1-yl)-1-phenylethanol derivatives.

Daniela de Vita , Luigi Scipione , Silvano Tortorella , Paolo Mellini , Barbara Di Rienzo , et al.
European Journal of Medicinal Chemistry, 2012, 49, pp.334-42. ⟨10.1016/j.ejmech.2012.01.034⟩
Journal articles pasteur-00968658v1
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New Promising Compounds with in Vitro Nanomolar Activity against Trypanosoma cruzi.

Laura Friggeri , Luigi Scipione , Roberta Costi , Marcel Kaiser , Francesca Moraca , et al.
ACS Medicinal Chemistry Letters, 2013, 4 (6), pp.538-41. ⟨10.1021/ml400039r⟩
Journal articles pasteur-01054197v1
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Identification of PR-SET7 and EZH2 selective inhibitors inducing cell death in human leukemia U937 cells.

Sergio Valente , Ilaria Lepore , Carmela Dell'Aversana , Maria Tardugno , Sabrina Castellano , et al.
Biochimie, 2012, 94 (11), pp.2308-13. ⟨10.1016/j.biochi.2012.06.003⟩
Journal articles pasteur-00968696v1