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Phenylpyrazolo[1,5-a]quinazolin-5(4H)-one: a suitable scaffold for the development of noncamptothecin topoisomerase I (Top1) inhibitors.
Sabrina Taliani
,
Isabella Pugliesi
,
Elisabetta Barresi
,
Silvia Salerno
,
Christophe Marchand
,
et al.
Journal articles
pasteur-00968854v1
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Quinolinonyl Non-Diketo Acid Derivatives as Inhibitors of HIV-1 Ribonuclease H and Polymerase Functions of Reverse Transcriptase
Antonella Messore
,
Angela Corona
,
Valentina Noemi Madia
,
Francesco Saccoliti
,
Valeria Tudino
,
et al.
Journal articles
hal-03831904v1
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New nucleotide-competitive non-nucleoside inhibitors of terminal deoxynucleotidyl transferase: discovery, characterization, and crystal structure in complex with the target.
Roberta Costi
,
Giuliana Cuzzucoli Crucitti
,
Luca Pescatori
,
Antonella Messore
,
Luigi Scipione
,
et al.
Journal articles
pasteur-00968827v1
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Effects of polyphenol compounds on influenza A virus replication and definition of their mechanism of action.
Rossella Fioravanti
,
Ignacio Celestino
,
Roberta Costi
,
Giuliana Cuzzucoli Crucitti
,
Luca Pescatori
,
et al.
Journal articles
pasteur-00968715v1
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6-(1-Benzyl-1H-pyrrol-2-yl)-2,4-dioxo-5-hexenoic acids as dual inhibitors of recombinant HIV-1 integrase and ribonuclease H, synthesized by a parallel synthesis approach.
Roberta Costi
,
Mathieu Métifiot
,
Francesca Esposito
,
Giuliana Cuzzucoli Crucitti
,
Luca Pescatori
,
et al.
Journal articles
pasteur-00968870v1
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Novel 3,5-bis(bromohydroxybenzylidene)piperidin-4-ones as coactivator-associated arginine methyltransferase 1 inhibitors: enzyme selectivity and cellular activity.
Donghang Cheng
,
Sergio Valente
,
Sabrina Castellano
,
Gianluca Sbardella
,
Roberto Di Santo
,
et al.
Journal articles
pasteur-00968654v1
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Pharmacophore assessment through 3-D QSAR: evaluation of the predictive ability on new derivatives by the application on a series of antitubercular agents.
Laura Friggeri
,
Flavio Ballante
,
Rino Ragno
,
Ira Musmuca
,
Daniela de Vita
,
et al.
Journal articles
pasteur-00968810v1
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Synthesis and antifungal activity of a new series of 2-(1H-imidazol-1-yl)-1-phenylethanol derivatives.
Daniela de Vita
,
Luigi Scipione
,
Silvano Tortorella
,
Paolo Mellini
,
Barbara Di Rienzo
,
et al.
Journal articles
pasteur-00968658v1
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New Promising Compounds with in Vitro Nanomolar Activity against Trypanosoma cruzi.
Laura Friggeri
,
Luigi Scipione
,
Roberta Costi
,
Marcel Kaiser
,
Francesca Moraca
,
et al.
Journal articles
pasteur-01054197v1
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Identification of PR-SET7 and EZH2 selective inhibitors inducing cell death in human leukemia U937 cells.
Sergio Valente
,
Ilaria Lepore
,
Carmela Dell'Aversana
,
Maria Tardugno
,
Sabrina Castellano
,
et al.
Journal articles
pasteur-00968696v1
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