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Discovery and pharmacological profile of new 1H-indazole-3-carboxamide and 2H-pyrrolo[3,4-c]quinoline derivatives as selective serotonin 4 receptor ligands.

Guido Furlotti , Maria Alessandra Alisi , Claudia Apicella , Alessandra Capezzone de Joannon , Nicola Cazzolla , et al.
Journal of Medicinal Chemistry, 2012, 55 (22), pp.9446-66. ⟨10.1021/jm300573d⟩
Journal articles pasteur-00968755v1

Quinolinonyl Non-Diketo Acid Derivatives as Inhibitors of HIV-1 Ribonuclease H and Polymerase Functions of Reverse Transcriptase

Antonella Messore , Angela Corona , Valentina Noemi Madia , Francesco Saccoliti , Valeria Tudino , et al.
Journal of Medicinal Chemistry, 2021, 64 (12), pp.8579-8598. ⟨10.1021/acs.jmedchem.1c00535⟩
Journal articles hal-03831904v1
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Novel 3,5-bis(bromohydroxybenzylidene)piperidin-4-ones as coactivator-associated arginine methyltransferase 1 inhibitors: enzyme selectivity and cellular activity.

Donghang Cheng , Sergio Valente , Sabrina Castellano , Gianluca Sbardella , Roberto Di Santo , et al.
Journal of Medicinal Chemistry, 2011, 54 (13), pp.4928-32. ⟨10.1021/jm200453n⟩
Journal articles pasteur-00968654v1
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Design, synthesis, and structure-activity relationship of N-arylnaphthylamine derivatives as amyloid aggregation inhibitors.

Roberto Di Santo , Roberta Costi , Giuliana Cuzzucoli Crucitti , Luca Pescatori , Federica Rosi , et al.
Journal of Medicinal Chemistry, 2012, 55 (19), pp.8538-48. ⟨10.1021/jm301105m⟩
Journal articles pasteur-00968739v1
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Pharmacophore assessment through 3-D QSAR: evaluation of the predictive ability on new derivatives by the application on a series of antitubercular agents.

Laura Friggeri , Flavio Ballante , Rino Ragno , Ira Musmuca , Daniela de Vita , et al.
Journal of Chemical Information and Modeling, 2013, 53 (6), pp.1463-74. ⟨10.1021/ci400132q⟩
Journal articles pasteur-00968810v1
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New Promising Compounds with in Vitro Nanomolar Activity against Trypanosoma cruzi.

Laura Friggeri , Luigi Scipione , Roberta Costi , Marcel Kaiser , Francesca Moraca , et al.
ACS Medicinal Chemistry Letters, 2013, 4 (6), pp.538-41. ⟨10.1021/ml400039r⟩
Journal articles pasteur-01054197v1
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Identification of PR-SET7 and EZH2 selective inhibitors inducing cell death in human leukemia U937 cells.

Sergio Valente , Ilaria Lepore , Carmela Dell'Aversana , Maria Tardugno , Sabrina Castellano , et al.
Biochimie, 2012, 94 (11), pp.2308-13. ⟨10.1016/j.biochi.2012.06.003⟩
Journal articles pasteur-00968696v1