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6-(1-Benzyl-1H-pyrrol-2-yl)-2,4-dioxo-5-hexenoic acids as dual inhibitors of recombinant HIV-1 integrase and ribonuclease H, synthesized by a parallel synthesis approach.

Roberta Costi , Mathieu Métifiot , Francesca Esposito , Giuliana Cuzzucoli Crucitti , Luca Pescatori , et al.
Journal of Medicinal Chemistry, 2013, 56 (21), pp.8588-98. ⟨10.1021/jm401040b⟩
Journal articles pasteur-00968870v1
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New nucleotide-competitive non-nucleoside inhibitors of terminal deoxynucleotidyl transferase: discovery, characterization, and crystal structure in complex with the target.

Roberta Costi , Giuliana Cuzzucoli Crucitti , Luca Pescatori , Antonella Messore , Luigi Scipione , et al.
Journal of Medicinal Chemistry, 2013, 56 (18), pp.7431-41. ⟨10.1021/jm4010187⟩
Journal articles pasteur-00968827v1

Quinolinonyl Non-Diketo Acid Derivatives as Inhibitors of HIV-1 Ribonuclease H and Polymerase Functions of Reverse Transcriptase

Antonella Messore , Angela Corona , Valentina Noemi Madia , Francesco Saccoliti , Valeria Tudino , et al.
Journal of Medicinal Chemistry, 2021, 64 (12), pp.8579-8598. ⟨10.1021/acs.jmedchem.1c00535⟩
Journal articles hal-03831904v1
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Design, synthesis, and structure-activity relationship of N-arylnaphthylamine derivatives as amyloid aggregation inhibitors.

Roberto Di Santo , Roberta Costi , Giuliana Cuzzucoli Crucitti , Luca Pescatori , Federica Rosi , et al.
Journal of Medicinal Chemistry, 2012, 55 (19), pp.8538-48. ⟨10.1021/jm301105m⟩
Journal articles pasteur-00968739v1
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Pharmacophore assessment through 3-D QSAR: evaluation of the predictive ability on new derivatives by the application on a series of antitubercular agents.

Laura Friggeri , Flavio Ballante , Rino Ragno , Ira Musmuca , Daniela de Vita , et al.
Journal of Chemical Information and Modeling, 2013, 53 (6), pp.1463-74. ⟨10.1021/ci400132q⟩
Journal articles pasteur-00968810v1
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New Promising Compounds with in Vitro Nanomolar Activity against Trypanosoma cruzi.

Laura Friggeri , Luigi Scipione , Roberta Costi , Marcel Kaiser , Francesca Moraca , et al.
ACS Medicinal Chemistry Letters, 2013, 4 (6), pp.538-41. ⟨10.1021/ml400039r⟩
Journal articles pasteur-01054197v1