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Structure: Internal structure identifier : 190928
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New nitrogen containing substituents at the indole-2-carboxamide yield high potent and broad spectrum indolylarylsulfone HIV-1 non-nucleoside reverse transcriptase inhibitors.

Giuseppe La Regina , Antonio Coluccia , Andrea Brancale , Francesco Piscitelli , Valeria Famiglini , et al.
Journal of Medicinal Chemistry, 2012, 55 (14), pp.6634-8. ⟨10.1021/jm300477h⟩
Journal articles pasteur-00969585v1
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Phenylpyrazolo[1,5-a]quinazolin-5(4H)-one: a suitable scaffold for the development of noncamptothecin topoisomerase I (Top1) inhibitors.

Sabrina Taliani , Isabella Pugliesi , Elisabetta Barresi , Silvia Salerno , Christophe Marchand , et al.
Journal of Medicinal Chemistry, 2013, 56 (18), pp.7458-62. ⟨10.1021/jm400932c⟩
Journal articles pasteur-00968854v1